Pipeline

Retatrutide: What We Know About Lilly's Next-Gen GLP-1

24% weight loss in Phase 2, three-hormone mechanism, and on track for FDA filing in 2026-2027. Here's what retatrutide actually is and why it matters.

April 5, 2026 · 6 min read

Bottom line

Retatrutide is Eli Lilly's next-generation weight-loss drug — a triple agonist targeting GLP-1, GIP, and glucagon. Phase 2 showed ~24% average weight loss at 48 weeks. Filing expected 2026-2027.

What triple agonist means

The glucagon piece adds fat oxidation and increased energy expenditure — where Zepbound turns down calorie intake, retatrutide also turns up calorie burn.

The numbers

Phase 2 TRIUMPH-1 at 48 weeks: 8.7% at 2mg, 17.1% at 4mg, 21.1% at 8mg, 24.2% at 12mg. Zepbound at 48 weeks was ~18%.

What we don't know

Long-term tolerability, maintenance dosing, launch price, cardiovascular outcomes data.

If you're on a GLP-1 today

Don't wait. Start with what's available. Retatrutide won't be broadly available until late 2026+. The weight-loss debt you accumulate waiting usually costs more than the switch difficulty later.